From: Low affinity glucocorticoid binding site ligands as potential anti-fibrogenics
Cold Competitor
IC50% (10-6 M)
dexamethasone
0.098 ± 0.003
progesterone
0.081 ± 0.010
clotrimazole
40 ± 12
metyrapone
310 ± 52
haloperidol
> 10000